From Mechanism-Based Retaining Glycosidase Inhibitors to Activity-Based Glycosidase Profiling-Reference-Cited by-同舟云学术

From Mechanism-Based Retaining Glycosidase Inhibitors to Activity-Based Glycosidase Profiling

Published:2024-08-30 Issue:36 Volume:146 Page:24729-24741
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Artola Marta¹^ORCID,Aerts Johannes M. F. G.¹^ORCID,van der Marel Gijsbert A.¹,Rovira Carme²³^ORCID,Codée Jeroen D. C.¹^ORCID,Davies Gideon J.⁴^ORCID,Overkleeft Herman S.¹^ORCID

Affiliation:

1. Leiden Institute of Chemistry, Leiden University, 2300 RA, Leiden, The Netherlands

2. Departament de Química Inorgànica I Orgànica & IQTCUB, Universitat de Barcelona, Barcelona 08028, Spain

3. Institució Catalana de Recerca i Estudis Avançats (ICREA), Barcelona 08020, Spain

4. Department of Chemistry, The University York, Heslington, York YO10 5DD, United Kingdom

Funder

Royal Society

Exacte en Natuurwetenschappen

Ministerio de Ciencia, Innovaci?n y Universidades

Ag?ncia de Gesti? d'Ajuts Universitaris i de Recerca

FP7 Ideas: European Research Council

University of Melbourne

H2020 European Research Council

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/jacs.4c08840

Reference82 articles.

1. Structural and sequence-based classification of glycoside hydrolases

2. The carbohydrate-active enzymes database (CAZy) in 2013

3. Catalytic mechanism of enzymic glycosyl transfer

4. STEREOCHEMISTRY AND THE MECHANISM OF ENZYMATIC REACTIONS

5. Compounds that react within the enzyme active site to form a covalent and irreversible bond, thereby irreversibly inactivating the enzyme, are sometimes referred to as ‘targeted covalent inhibitors’, ‘suicide inhibitors’ or ‘activity-based inhibitors’. In line with other practitioners in the field (see also the titles of some of the references below) we have chosen to use the term ‘mechanism-based inhibitors’, which is also the term recommended by IUPAC. See also https://iupac.qmul.ac.uk/gtpoc/M.html.