Synthesis and biological activity of novel bis-indole inhibitors of bacterial transcription initiation complex formation-Reference-Cited by-同舟云学术

Synthesis and biological activity of novel bis-indole inhibitors of bacterial transcription initiation complex formation

Published:2014 Issue:18 Volume:12 Page:2882-2894
ISSN:1477-0520
Container-title:Org. Biomol. Chem.
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Mielczarek Marcin¹²³,Devakaram Ruth V.¹²³,Ma Cong⁴⁵⁶,Yang Xiao⁴⁵⁶,Kandemir Hakan¹²³,Purwono Bambang¹²³,Black David StC.¹²³,Griffith Renate⁷⁸²³,Lewis Peter J.⁴⁵⁶,Kumar Naresh¹²³

Affiliation:

1. School of Chemistry

2. The University of New South Wales

3. Sydney, Australia

4. School of Environmental and Life Sciences

5. University of Newcastle

6. Callaghan, Australia

7. School of Medical Sciences

8. Department of Pharmacology

Abstract

The synthesis of novel bis-indole amides and glyoxylamides as bacterial transcription complex formation inhibitors and their structure–activity relationships are discussed.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/OB/C4OB00460D

Reference32 articles.

1. Antibiotic resistance: an increasing problem?

2. Antibiotic resistance in microbes

3. Antimicrobial Resistance and Aging: Beginning of the End of the Antibiotic Era?

4. Antibiotic and biocide resistance in bacteria: Introduction

5. Antibiotic resistance in Gram-positive bacteria: epidemiological aspects

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