Facile one-pot synthesis of 2-amino-1,3,4-oxadiazole tethered peptidomimetics by molecular-iodine-mediated cyclodeselenization-Reference-Cited by-同舟云学术

Facile one-pot synthesis of 2-amino-1,3,4-oxadiazole tethered peptidomimetics by molecular-iodine-mediated cyclodeselenization

Published:2017 Issue:19 Volume:41 Page:11225-11229
ISSN:1144-0546
Container-title:New Journal of Chemistry
language:en
Short-container-title:New J. Chem.

Author:

Santhosh L.¹²³⁴⁵,Srinivasulu C.¹²³⁴⁵,Durgamma S.¹²³⁴⁵,Prabhu Girish¹²³⁴⁵,Sureshbabu Vommina V.¹²³⁴⁵^ORCID

Affiliation:

1. Peptide Research Laboratory

2. Department of Studies in Chemistry

3. Central College Campus

4. Dr B. R. AmbedkarVeedhi

5. Bangalore University

Abstract

Mild and highly efficient I₂ and Et₃N aided cyclodeselenization of in situ generated selenosemicarbazide is described to obtain 2-amino-1,3,4-oxadiazole peptidomimetics.

Funder

Science and Engineering Research Board

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,General Chemistry,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2017/NJ/C7NJ02278F

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5. Discovery of novel antitubercular 1,5-dimethyl-2-phenyl-4-([5-(arylamino)-1,3,4-oxadiazol-2-yl]methylamino)-1,2-dihydro-3H-pyrazol-3-one analogues

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