Highly diastereoselective crystallization-induced asymmetric transformation of 1,3-disubstituted-tetrahydro-β-carbolines in water-Reference-Cited by-同舟云学术

Highly diastereoselective crystallization-induced asymmetric transformation of 1,3-disubstituted-tetrahydro-β-carbolines in water

Published:2017 Issue:75 Volume:7 Page:47753-47757
ISSN:2046-2069
Container-title:RSC Adv.
language:en
Short-container-title:RSC Adv.

Author:

Meng Tian-Zhuo¹²³⁴⁵,Shi Xiao-Xin¹²³⁴⁵^ORCID,Qu Hui-Ya¹²³⁴⁵,Zhang Yi¹²³⁴⁵,Huang Zhong-Shou¹²³⁴⁵,Fan Qi-Qi¹²³⁴⁵

Affiliation:

1. Department of Pharmaceutical Engineering

2. School of Pharmacy

3. East China University of Science and Technology

4. Shanghai 200237

5. P. R. China

Abstract

A green and highly stereoselective method for the synthesis of cis or trans-1,3-disubstituted-tetrahydro-β-carbolines has been developed using water as the solvent.

Funder

National Natural Science Foundation of China

Shanghai Educational Development Foundation

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/RA/C7RA08811F

Reference76 articles.

1. The E factor 25 years on: the rise of green chemistry and sustainability

2. Overcoming barriers to green chemistry in the pharmaceutical industry – the Green Aspiration Level™ concept

3. Fundamentals of green chemistry: efficiency in reaction design

4. Chemistry: It's not easy being green

5. Green Chemistry: Principles and Practice

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