Chemical probes and inhibitors of bromodomains outside the BET family-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Chemical probes and inhibitors of bromodomains outside the BET family

Published:2016 Issue:12 Volume:7 Page:2246-2264
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Moustakim Moses¹²³⁴⁵^ORCID,Clark Peter G. K.¹⁶⁷⁸,Hay Duncan A.⁹¹⁰⁴,Dixon Darren J.¹²³⁴,Brennan Paul E.⁵²⁴¹¹¹²

Affiliation:

1. Department of Chemistry

2. University of Oxford

3. Oxford OX1 3TA

4. UK

5. Structural Genomics Consortium

6. Simon Fraser University

7. Burnaby V5A 1S6

8. Canada

9. Evotec (UK) Ltd

10. Oxfordshire OX14 4RZ

11. Target Discovery Institute

12. Nuffield Department of Medicine

Abstract

Significant progress has been made in discovering inhibitors and chemical probes of bromodomains, epigenetic readers of lysine acetylation.

Funder

Wellcome Trust

Engineering and Physical Sciences Research Council

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/MD/C6MD00373G

Reference121 articles.

1. Epigenetic protein families: a new frontier for drug discovery

2. Epigenetics in Cancer

3. Cancer-epigenetics comes of age

4. Targeting Epigenetic Readers in Cancer

5. Role of Epigenetics in Inflammation-Associated Diseases

Cited by 53 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Targeting Bromodomain-Containing Protein 9 in Human Uterine Fibroid Cells;Reproductive Sciences;2024-06-10

2. Bromodomain-Containing Protein 9 Regulates Signaling Pathways and Reprograms the Epigenome in Immortalized Human Uterine Fibroid Cells;International Journal of Molecular Sciences;2024-01-11

3. Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3;Bioorganic & Medicinal Chemistry Letters;2024-01

4. Targeting Epigenetic Readers Using Small Molecule Binders and PROTAC Degraders;Interdisciplinary Cancer Research;2024

5. BET Bromodomain Inhibitors as an Emerging Class of Anticancer Agents;Handbook of Cancer and Immunology;2023-11-08

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3