Synthesis of isoxazolidine-containing uridine derivatives as caprazamycin analogues
Author:
Affiliation:
1. Faculty of Pharmaceutical Sciences
2. Hokkaido University
3. Sapporo 060-0812
4. Japan
5. Center for Research and Education on Drug Discovery
Abstract
Simplification of caprazamycins was conducted by scaffold-hopping of the structurally complex diazepanone moiety to the isoxazolidine scaffold.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB02142H
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