Multivalent ligands for the serotonin 5-HT4 receptor-Reference-Cited by-同舟云学术

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Multivalent ligands for the serotonin 5-HT4 receptor

Published:2017 Issue:3 Volume:8 Page:647-651
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Castriconi Federica¹²³⁴⁵,Paolino Marco¹²³⁴⁵,Donati Alessandro¹²³⁴⁵,Giuliani Germano¹²³⁴⁵,Anzini Maurizio¹²³⁴⁵,Mennuni Laura⁶⁷⁵,Sabatini Chiara⁶⁷⁵,Lanza Marco⁶⁷⁵,Caselli Gianfranco⁶⁷⁵,Makovec Francesco⁶⁷⁵,Sbraccia Maria⁸⁹¹⁰⁵,Molinari Paola⁸⁹¹⁰⁵,Costa Tommaso⁸⁹¹⁰⁵,Cappelli Andrea¹²³⁴⁵^ORCID

Affiliation:

1. Dipartimento di Biotecnologie

2. Chimica e Farmacia and European Research Centre for Drug Discovery and Development

3. Università degli Studi di Siena

4. 53100 Siena

5. Italy

6. Rottapharm Biotech S.r.l.

7. 20900 Monza

8. Dipartimento di Farmacologia

9. Istituto Superiore di Sanità

10. 00161 Roma

Abstract

Multivalency does not improve the binding and functional activities of ML10302 at 5-HT₄ receptors.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/MD/C6MD00458J

Reference22 articles.

1. Molecular biology of 5-HT receptors

2. Serotonin Receptors

3. The gastrointestinal prokinetic benzamide derivatives are agonists at the non-classical 5-HT receptor (5-HT4) positively coupled to adenylate cyclase in neurons

4. 5-HT4 receptors: History, molecular pharmacology and brain functions

5. 5-HT4 Receptor Ligands: Applications and New Prospects

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2. Covalent hyaluronic-based coating of magnetite nanoparticles: Preparation, physicochemical and biological characterization;Materials Science and Engineering: C;2020-02

3. 2016 Philip S. Portoghese Medicinal Chemistry Lectureship: Designing Bivalent or Bitopic Molecules for G-Protein Coupled Receptors. The Whole Is Greater Than the Sum of Its Parts;Journal of Medicinal Chemistry;2019-09-09

4. ML10302;Reference Module in Biomedical Sciences;2018

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