The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies-Reference-Cited by-同舟云学术

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The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies

Published:2016 Issue:21 Volume:14 Page:4853-4858
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Di Fiore Anna¹²³,De Simone Giuseppina¹²³,Alterio Vincenzo¹²³,Riccio Vincenzo¹²³,Winum Jean-Yves⁴⁵⁶⁷⁸,Carta Fabrizio⁹¹⁰¹¹¹²³,Supuran Claudiu T.⁹¹⁰¹¹¹²³

Affiliation:

1. Istituto di Biostrutture e Bioimmagini-CNR

2. 80134 Napoli

3. Italy

4. Institut des Biomolécules Max Mousseron (IBMM) UMR 5247 CNRS

5. ENSCM

6. Université de Montpellier

7. Bâtiment de Recherche Max Mousseron

8. Ecole Nationale Supérieure de Chimie de Montpellier

9. Università degli Studi di Firenze

10. Polo Scientifico

11. Laboratorio di Chimica Bioinorganica

12. 50019 Sesto Fiorentino

Abstract

Inhibition and X-ray crystallographic data for the binding of JNJ-26990990 and its S,S-dioxide analog to hCAs have been reported.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB00803H

Reference43 articles.

1. Novel, Broad-Spectrum Anticonvulsants Containing a Sulfamide Group: Advancement of N-((Benzo[b]thien-3-yl)methyl)sulfamide (JNJ-26990990) into Human Clinical Studies

2. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

3. Antiepileptic activity of zonisamide on hippocampal CA3 neurons does not depend on carbonic anhydrase inhibition

4. Molecular modeling study for the binding of zonisamide and topiramate to the human mitochondrial carbonic anhydrase isoform VA

5. Anticonvulsant O-alkyl sulfamates. 2,3:4,5-Bis-O-(1-methylethylidene)-.beta.-D-fructopyranose sulfamate and related compounds

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