A facile one pot route for the synthesis of imide tethered peptidomimetics-Reference-Cited by-同舟云学术

A facile one pot route for the synthesis of imide tethered peptidomimetics

Published:2016 Issue:2 Volume:14 Page:556-563
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Panduranga Veladi¹²³⁴,Prabhu Girish¹²³⁴,Kumar Roopesh¹²³⁴,Basavaprabhu Basavaprabhu¹²³⁴,Sureshbabu Vommina V.¹²³⁴

Affiliation:

1. Peptide Research Laboratory

2. Department of Studies in Chemistry

3. Bangalore 560 001

4. India

Abstract

A simple and efficient method for the synthesis of N,N’-orthogonally protected imide tethered peptidomimetics is presented. The imide peptidomimetics were synthesized by coupling the in situ generated selenocarboxylate of N^α-protected amino acids with N^α-protected amino acid azides in good yields.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C5OB01708D

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