Determination of the absolute configuration of phosphinic analogues of glutamate-Reference-Cited by-同舟云学术

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Determination of the absolute configuration of phosphinic analogues of glutamate

Published:2015 Issue:4 Volume:13 Page:1106-1112
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Commare Bruno¹²³⁴⁵,Rigault Delphine¹²³⁴⁵,Lemasson Isabelle A.¹²³⁴⁵,Deschamps Patrick⁶⁷³⁸⁹,Tomas Alain⁶⁷³⁸⁹,Roussel Pascal¹⁰¹¹¹²⁹,Brabet Isabelle¹³¹⁴¹⁵¹⁶⁹,Goudet Cyril¹³¹⁴¹⁵¹⁶⁹,Pin Jean-Philippe¹³¹⁴¹⁵¹⁶⁹,Leroux Frédéric R.¹⁷¹⁸¹⁹²⁰⁹,Colobert Françoise¹⁷¹⁸¹⁹²⁰⁹,Acher Francine C.¹²³⁴⁵

Affiliation:

1. Laboratoire de Chimie & Biochimie Pharmacologiques et Toxicologiques

2. UMR CNRS 8601

3. Université Paris Descartes

4. Sorbonne Paris Cité

5. Paris cedex 06

6. Laboratoire de Cristallographie et RMN Biologiques

7. UMR CNRS 8015

8. 75270 Paris cedex 06

9. France

10. Unité de Catalyse et Chimie du solide

11. UMR CNRS 8012

12. École Nationale Supérieure de Chimie de Lille BP 90108-59652 Villeneuve d'Ascq cedex

13. Institut de Génomique Fonctionnelle

14. Centre National de la Recherche Scientifique Unité Mixte de Recherche 5203

15. Université de Montpellier

16. F-34094 Montpellier

17. Laboratoire de Chimie Moléculaire

18. UMR CNRS 7509

19. Université de Strasbourg

20. Strasbourg

Abstract

Stereomers of LSP1-2111 have been separated, their absolute configuration and agonist activity at mGlu4R determined.

Funder

Agence Nationale de la Recherche

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB01960A

Reference33 articles.

1. Design, Synthesis, and Activity of Analogues of Phosphinothricin as Inhibitors of Glutamine Synthetase

2. Phosphinothricin Analogues as Inhibitors of Plant Glutamine Synthetases

3. Remarkable Potential of the α-Aminophosphonate/Phosphinate Structural Motif in Medicinal Chemistry

4. N-substituted aminomethanephosphonic and aminomethane-P-methylphosphinic acids as inhibitors of ureases

5. Identification of very potent inhibitor of human aminopeptidase N (CD13)

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1. Organoaluminum Reagents;Reference Module in Chemistry, Molecular Sciences and Chemical Engineering;2024

2. International Union of Basic and Clinical Pharmacology. CXI. Pharmacology, Signaling, and Physiology of Metabotropic Glutamate Receptors;Pharmacological Reviews;2020-12-23

3. From Industrial Method to the Use of Silylated P(III) Reagents for the Synthesis of Relevant Phosphonylated Molecules;Organic Process Research & Development;2020-01-23

4. Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites;Journal of Medicinal Chemistry;2018-02-04

5. Phosphonic acid: preparation and applications;Beilstein Journal of Organic Chemistry;2017-10-20

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