A convenient approach to an advanced intermediate toward the naturally occurring, bioactive 6-substituted 5-hydroxy-4-aryl-1H-quinolin-2-ones
Author:
Affiliation:
1. Instituto de Química Rosario (IQUIR
2. CONICET-UNR) and Facultad de Ciencias Bioquímicas y Farmacéuticas
3. Universidad Nacional de Rosario
4. S2002LRK Rosario
5. Argentina
Abstract
An advanced intermediate for the total synthesis of the 5-hydroxy-4-aryl-3,4-dihydro-1H-quinolin-2-one natural products and a 3,4-bisdesoxy analog of peniprequinolone were synthesized.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/OB/C5OB02680F
Reference120 articles.
1. Privileged Structures: Applications in Drug Discovery
2. The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
3. A. Méndez-Vilas , Science Against Microbial Pathogens: Communicating Current Research and Technological Advances, Formatex, Badajoz, Spain, 2011, vol. 2
4. The concept of privileged structures in rational drug design: focus on acridine and quinoline scaffolds in neurodegenerative and protozoan diseases
5. Quinoline as a Privileged Scaffold in Cancer Drug Discovery
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