Preparation, anti-trypanosomal activity and localisation of a series of dipeptide-based vinyl sulfones-Reference-Cited by-同舟云学术

Preparation, anti-trypanosomal activity and localisation of a series of dipeptide-based vinyl sulfones

Published:2014 Issue:38 Volume:12 Page:7561-7571
ISSN:1477-0520
Container-title:Org. Biomol. Chem.
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Doherty William¹²³⁴,James Jinju¹²³⁴,Evans Paul¹²³⁴,Martin Laura⁵⁶⁷⁸,Adler Nikoletta⁵⁶⁷⁸,Nolan Derek⁵⁶⁷⁸,Knox Andrew⁵⁶⁷⁸

Affiliation:

1. Centre for Synthesis and Chemical Biology

2. School of Chemistry and Chemical Biology

3. University College Dublin

4. Dublin 4, Ireland

5. School of Biochemistry and Immunology

6. Trinity Biomedical Sciences Institute

7. Trinity College Dublin

8. Dublin 2, Ireland

Abstract

An improved, Weinreb amide-based, synthesis of anti-trypanosomal lysine-containing vinyl sulfones is described incorporating, as a feature, diversity at the ε-lysine amino group.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/OB/C4OB01412J

Reference48 articles.

1. The chemistry of vinyl sulphones

2. Multiply convergent syntheses via conjugate-addition reactions to cycloalkenyl sulfones

3. Evolving Organic Synthesis Fostered by the Pluripotent Phenylsulfone Moiety

4. The Use of Sulfonyl 1,3-Dienes in Organic Synthesis

5. Vinyl sulfones: Synthetic preparations and medicinal chemistry applications

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