Synthesis of benzo[1,3]oxazines via copper(i)-catalyzed cascade annulation of nitriles, aldehydes and diaryliodonium salts-Reference-Cited by-同舟云学术

Synthesis of benzo[1,3]oxazines via copper(i)-catalyzed cascade annulation of nitriles, aldehydes and diaryliodonium salts

Published:2016 Issue:4 Volume:3 Page:501-504
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Sheng Jinyu¹²³⁴⁵,Su Xiang¹²³⁴⁵,Cao Chengyao¹²³⁴⁵,Chen Chao¹²³⁴⁵

Affiliation:

1. Key Laboratory of Bioorganic Phosphorus Chemistry & Chemical Biology (Ministry of Education)

2. Department of Chemistry

3. Tsinghua University

4. Beijing 100084

5. China

Abstract

A copper(i)-catalyzed one-pot [2 + 2 + 2] cascade annulation reaction of diaryliodoniums, nitriles, and aldehydes has been developed for the efficient synthesis of 2,4-substituted benzoxazine derivatives.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/QO/C6QO00012F

Reference58 articles.

1. The Leupyrrins: A Structurally Unique Family of Secondary Metabolites from the Myxobacterium Sorangium cellulosum#

2. Potent, Novel in Vitro Inhibitors of the Pseudomonas aeruginosa Deacetylase LpxC

3. High-Throughput Catch-and-Release Synthesis of Oxazoline Hydroxamates. Structure−Activity Relationships in Novel Inhibitors of Escherichia coli LpxC: In Vitro Enzyme Inhibition and Antibacterial Properties

4. Oxoazabenzo[de]anthracenes Conjugated to Amino Acids: Synthesis and Evaluation as DNA-Binding Antitumor Agents

5. Design and synthesis of 4H-3,1-benzoxazin-4-ones as potent alternate substrate inhibitors of human leukocyte elastase

Cited by 29 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. 4H-3,1-Benzoxazines and their dihydro derivatives: synthesis, reactivity, and biological activity;Russian Chemical Bulletin;2024-05

2. Copper-Catalyzed Synthesis of Quinoline-4-thiols from Diaryliodonium Salts, Alkynyl Sulfides, and Nitriles;Organic Letters;2023-07-13

3. Synthesis of 1-Tosylspiro[3,1-benzoxazine-4,1′-cycloalkan]-2-imines;Russian Journal of Organic Chemistry;2022-10

4. Diaryliodonium(iii) salts in one-pot double functionalization of C–I^III and ortho C–H bonds;Organic & Biomolecular Chemistry;2022

5. Cu-catalyzed [2 + 2 + 1] cascade annulation of vinyl iodonium salts with elemental sulfur/selenium for the modular synthesis of thiophenes and selenophenes;New Journal of Chemistry;2022