A silver-promoted solid-phase guanidylation process enables the first total synthesis of stictamide A-Reference-Cited by-同舟云学术

A silver-promoted solid-phase guanidylation process enables the first total synthesis of stictamide A

Published:2015 Issue:115 Volume:5 Page:94654-94657
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Li Xiang¹²³⁴⁵,Li Yu-lei¹²³⁴⁵,Chen Yan⁶⁷⁸⁵,Zou Yan¹²³⁴⁵,Zhuo Xiao-bin¹²³⁴⁵,Wu Qiu-ye¹²³⁴⁵,Zhao Qing-jie¹²³⁴⁵,Hu Hong-gang¹²³⁴⁵

Affiliation:

1. Department of Organic Chemistry

2. School of Pharmacy

3. Second Military Medical University

4. Shanghai 200433

5. China

6. Department of Pharmacy

7. General Hospital of Beijing Military Region

8. Beijing 100700

Abstract

First total synthesis of stictamide A, a structurally unique peptide with a statine motif and a N-prenyl modified arginine in the side chain, is disclosed with a novel silver-promoted solid-phase strategy for the first time.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA20976E

Reference43 articles.

1. Highly active and selective endopeptidases with programmed substrate specificities

2. Cell attachment activity of fibronectin can be duplicated by small synthetic fragments of the molecule

3. Selective RGD-Mediated Adhesion of Osteoblasts at Surfaces of Implants

4. Exploration of Cyanine Compounds as Selective Inhibitors of Protein Arginine Methyltransferases: Synthesis and Biological Evaluation

5. A Versatile One-Pot Synthesis of 1,3-Substituted Guanidines from Carbamoyl Isothiocyanates

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Microwave-Assisted Solid Phase Synthesis of Different Peptide Bonds: Recent Advancements;Current Microwave Chemistry;2023-09

2. Silver-promoted solid-phase guanidinylation enables the first synthesis of arginine glycosylated Samoamide A cyclopeptide analogue;Frontiers in Chemistry;2023-01-04

3. A toolbox of diverse arginine N-glycosylated peptides and specific antibodies;Bioorganic Chemistry;2023-01

4. Highly stereoselective multigram scale synthesis of (3S,4S)-Statine and (3S,4S)-N-Benzylstatine;Results in Chemistry;2022-01

5. Diastereoselective Synthesis of (–)-Bestatin, Epibestatin, Phebestin and (3S,4R)-4-Amino-3-hydroxy-5-phenylpentanoic Acid from an Aldehyde Derived from d-Phenylalanine;SynOpen;2019-10