Metal-free oxidative cyclization of trifluoroacetimidohydrazides with methylhetarenes: a facile access to 3-hetaryl-5-trifluoromethyl-1,2,4-triazoles-Reference-Cited by-同舟云学术

Metal-free oxidative cyclization of trifluoroacetimidohydrazides with methylhetarenes: a facile access to 3-hetaryl-5-trifluoromethyl-1,2,4-triazoles

Published:2021 Issue:16 Volume:8 Page:4490-4495
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Zhang Jiajun¹²³⁴⁵,Xu Tian-Hui¹²³⁴⁵,Chen Zhengkai¹²³⁴⁵^ORCID,Wu Xiao-Feng⁶⁷⁸⁹¹⁰^ORCID

Affiliation:

1. Department of Chemistry

2. Key Laboratory of Surface & Interface Science of Polymer Materials of Zhejiang Province

3. Zhejiang Sci-Tech University

4. Hangzhou 310018

5. People's Republic of China

6. Dalian National Laboratory for Clean Energy

7. Dalian Institute of Chemical Physics

8. Chinese Academy of Sciences

9. Dalian 116023

10. China

Abstract

A metal-free oxidative cyclization of trifluoroacetimidohydrazides with methylhetarenes for the efficient synthesis of 3-hetaryl-5-trifluoromethyl-1,2,4-triazoles has been developed.

Funder

Natural Science Foundation of Zhejiang Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/QO/D1QO00790D

Reference50 articles.

1. Synthesis and Pharmacological Activity of Triazole Derivatives Inhibiting Eosinophilia

2. New bis-aminomercaptotriazoles and bis-triazolothiadiazoles as possible anticancer agents

3. Synthesis and Antitumor Activity of 1,5-Disubstituted 1,2,4-Triazoles as Cis-Restricted Combretastatin Analogues

4. Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4H-1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors

5. Synthesis, Antimitotic and Antivascular Activity of 1-(3′,4′,5′-Trimethoxybenzoyl)-3-arylamino-5-amino-1,2,4-triazoles

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