Triarylethylene-indolin-2,3-dione molecular conjugates: design, synthesis, docking studies and anti-proliferation evaluation-Reference-Cited by-同舟云学术

Triarylethylene-indolin-2,3-dione molecular conjugates: design, synthesis, docking studies and anti-proliferation evaluation

Published:2019 Issue:72 Volume:9 Page:42409-42414
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Kumar Sumit¹²³⁴,Palma Gabriella⁵⁶⁷⁸,Perumal Shanen⁵⁶⁷⁸^ORCID,Kaur Mandeep⁵⁶⁷⁸,Singh-Pillay Ashona⁹¹⁰¹¹⁸,Raj Raghu¹¹²¹³⁴,Singh Parvesh⁹¹⁰¹¹⁸,Kumar Vipan¹²³⁴^ORCID

Affiliation:

1. Department of Chemistry

2. Guru Nanak Dev University

3. Amritsar-143005

4. India

5. School of Molecular and Cell Biology

6. University of the Witswatersrand

7. Johannesburg

8. South Africa

9. School of Chemistry and Physics

10. University of KwaZulu Natal

11. Durban 4000

12. DAV College

13. Amritsar-143001

Abstract

A series of 1H-1,2,3-triazole-linked ospemifene–isatin and O-methylated ospemifene–isatin conjugates were synthesized and assayed for their anti-proliferative activities against estrogen-responsive as well as estrogen-non-responsive cells.

Funder

Science and Engineering Research Board

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/RA/C9RA08776A

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