Organocatalytic asymmetric [4+2] cyclization of 2-benzothiazolimines with azlactones: access to chiral benzothiazolopyrimidine derivatives-Reference-Cited by-同舟云学术

Organocatalytic asymmetric [4+2] cyclization of 2-benzothiazolimines with azlactones: access to chiral benzothiazolopyrimidine derivatives

Published:2020 Issue:21 Volume:56 Page:3155-3158
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Ni Qijian¹²³⁴⁵^ORCID,Wang Xuyang¹²³⁴⁵,Xu Fangfang¹²³⁴⁵,Chen Xiaoyun⁶⁷⁸⁹^ORCID,Song Xiaoxiao¹²³⁴⁵^ORCID

Affiliation:

1. College of Chemistry and Materials Science

2. Key Laboratory of Functionalized Molecular Solids

3. Ministry of Education

4. Anhui Laboratory of Molecule-Based Materials

5. Anhui Normal University

6. School of Environmental and Chemical Engineering

7. Jiangsu University of Science and Technology

8. Zhenjiang

9. P. R. China

Abstract

A squaramide catalyzed regiospecific and stereoselective [4+2] cyclization of 2-benzothiazolimines with azlactones has been established.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Anhui Province

Excellent Young Talents Fund Program of Higher Education Institutions of Anhui Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2020/CC/D0CC00736F

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2. In vitro Activity and Safety Assessment of New Synthesized Thiazolo Pyrimidine Derivatives Augmented with Albendazole against Echinococcus Multilocularis Metacestodes in Balb/C Mice

3. Chem-bioinformatics and in vitro approaches for candidate optimization: a case study of NSC745689 as a promising antitumor agent

4. Identification of an allosteric benzothiazolopyrimidone inhibitor of the oncogenic protein tyrosine phosphatase SHP2

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