5-(Methylthio)tetrazoles as versatile synthons in the stereoselective synthesis of polycyclic pyrazolines via photoinduced intramolecular nitrile imine–alkene 1,3-dipolar cycloaddition-Reference-Cited by-同舟云学术

5-(Methylthio)tetrazoles as versatile synthons in the stereoselective synthesis of polycyclic pyrazolines via photoinduced intramolecular nitrile imine–alkene 1,3-dipolar cycloaddition

Published:2014 Issue:6 Volume:5 Page:2407-2415
ISSN:2041-6520
Container-title:Chem. Sci.
language:en
Short-container-title:Chem. Sci.

Author:

Pla Daniel¹²³,Tan Derek S.¹²³⁴²,Gin David Y.¹²³⁴²

Affiliation:

1. Molecular Pharmacology and Chemistry Program

2. Memorial Sloan-Kettering Cancer Center

3. New York, USA

4. Tri-Institutional Research Program

Abstract

A versatile thioether substituent on tetrazoles enables facile photoinduced intramolecular nitrile imine cycloadditions to form polycyclic pyrazolines.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/SC/C4SC00107A

Reference73 articles.

1. Synthesis and Biological Activity of Chiral Dihydropyrazole: Potential Lead for Drug Design

2. Biological Activities of Pyrazoline Derivatives -A Recent Development

3. Recent Advances in the Chemistry of Pyrazoles. Properties, Biological Activities, and Syntheses

4. J. T. Sharp , in Synthetic Applications of 1,3-Dipolar Cycloaddition Chemistry toward Heterocycles and Natural Products, ed. A. Padwa and W. H. Pearson, Wiley, New York, 2002, ch. 7, pp. 473–537

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