Metal-free approach for hindered amide-bond formation with hypervalent iodine(iii) reagents: application to hindered peptide synthesis
Author:
Affiliation:
1. Graduate School of Pharmaceutical Sciences
2. Kyoto University
3. Kyoto 606-8501
4. Japan
5. Fukui Institute for Fundamental Chemistry
6. Kyoto 606-8103
7. School of Chemical Engineering and Light Industry
Abstract
A new, bulky amide and peptide synthesis with hypervalent iodine(iii) reagent/pyridine–hydrogen fluoride complex under mild and metal-free conditions was developed by using α-amino esters with potential activating group (PAG) at the ester residue.
Funder
Japan Society for the Promotion of Science
Publisher
Royal Society of Chemistry (RSC)
Subject
Pollution,Environmental Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2021/GC/D0GC03912H
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