Facile access to N-formyl imide as an N-formylating agent for the direct synthesis of N-formamides, benzimidazoles and quinazolinones-Reference-Cited by-同舟云学术

Facile access to N-formyl imide as an N-formylating agent for the direct synthesis of N-formamides, benzimidazoles and quinazolinones

Published:2020 Issue:29 Volume:18 Page:5726-5733
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Huang Hsin-Yi¹²³⁴,Lin Xiu-Yi¹²³⁴,Yen Shih-Yao¹²³⁴,Liang Chien-Fu¹²³⁴^ORCID

Affiliation:

1. Department of Chemistry

2. National Chung Hsing University

3. Taichung

4. Taiwan

Abstract

We developed a green method to produce N-formyl imides using acylamidines in water. Subsequently, N-formyl imide can be as a new water-tolerant N-formylating agent for the synthesis of N-formamides, benzimidazoles and quinazolinones.

Funder

Ministry of Science and Technology, Taiwan

National Chung-Hsing University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/D0OB01080D

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