NMR-based platform for fragment-based lead discovery used in screening BRD4-targeted compounds-Reference-Cited by-同舟云学术

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NMR-based platform for fragment-based lead discovery used in screening BRD4-targeted compounds

Published:2016-05-30 Issue:7 Volume:37 Page:984-993
ISSN:1671-4083
Container-title:Acta Pharmacologica Sinica
language:en
Short-container-title:Acta Pharmacol Sin

Author:

Yu Jun-lan,Chen Tian-tian,Zhou Chen,Lian Fu-lin,Tang Xu-long,Wen Yi,Shen Jing-kang,Xu Ye-chun,Xiong Bing,Zhang Nai-xia

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Pharmacology,General Medicine

Link

http://www.nature.com/articles/aps201619.pdf

Reference45 articles.

1. Erlanson DA . Introduction to fragment-based drug discovery. Top Curr Chem 2012; 317: 1–32.

2. Congreve M, Chessari G, Tisi D, Woodhead AJ . Recent developments in fragment-based drug discovery. J Med Chem 2008; 51: 3661–80.

3. Hanzawa H, Takizawa T . NMR in the fragment-based drug discovery. Tanpakushitsu Kakusan Koso 2009; 54 (12 Suppl): 1617–21. Japanese.

4. Harner MJ, Frank AO, Fesik SW . Fragment-based drug discovery using NMR spectroscopy. J Biomol NMR 2013; 56: 65–75.

5. Campos-Olivas R . NMR screening and hit validation in fragment based drug discovery. Curr Top Med Chem 2011; 11: 43–67.

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