General access to cubanes as benzene bioisosteres-Reference-Cited by-同舟云学术

General access to cubanes as benzene bioisosteres

Published:2023-04-04 Issue:7965 Volume:618 Page:513-518
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Wiesenfeldt Mario P.,Rossi-Ashton James A.,Perry Ian B.,Diesel Johannes,Garry Olivia L.,Bartels Florian^ORCID,Coote Susannah C.^ORCID,Ma Xiaoshen,Yeung Charles S.,Bennett David J.^ORCID,MacMillan David W. C.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

https://www.nature.com/articles/s41586-023-06021-8.pdf

Reference49 articles.

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2. Mykhailiuk, P. K. Saturated bioisosteres of benzene: where to go next? Org. Biomol. Chem. 17, 2839–2849 (2019).

3. Stepan, A. F. et al. Application of the bicyclo[1.1.1]pentane motif as a nonclassical phenyl ring bioisostere in the design of a potent and orally active γ-secretase inhibitor. J. Med. Chem. 55, 3414–3424 (2012).

4. Gianatassio, R. et al. Strain-release amination. Science 351, 241–246 (2016).

5. Zhang, X. et al. Copper-mediated synthesis of drug-like bicyclopentanes. Nature 580, 220–226 (2020).

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