Occupancy of dopamine D2 and D3 receptors by a novel D3 partial agonist BP1.4979: a [11C]-(+)-PHNO PET study in humans-Reference-Cited by-同舟云学术

Occupancy of dopamine D2 and D3 receptors by a novel D3 partial agonist BP1.4979: a [11C]-(+)-PHNO PET study in humans

Published:2018-11-30 Issue:7 Volume:44 Page:1284-1290
ISSN:0893-133X
Container-title:Neuropsychopharmacology
language:en
Short-container-title:Neuropsychopharmacol.

Author:

Di Ciano Patricia,Mansouri Esmaeil,Tong Junchao,Wilson Alan A.,Houle Sylvain,Boileau Isabelle,Duvauchelle Thierry,Robert Philippe,Schwartz Jean Charles,Le Foll Bernard

Funder

Bioprojet

Publisher

Springer Science and Business Media LLC

Subject

Psychiatry and Mental health,Pharmacology

Link

http://www.nature.com/articles/s41386-018-0285-4.pdf

Reference29 articles.

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3. Sokoloff P, Giros B, Martres MP, Bouthenet ML, Schwartz JC. Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics. Nature. 1990;347:146–51.

4. Heidbreder C. Rationale in support of the use of selective dopamine D(3) receptor antagonists for the pharmacotherapeutic management of substance use disorders. Naunyn Schmiede Arch Pharmacol. 2013;386:167–76.

5. Sibley DR, Monsma FJ. Molecular biology of dopamine receptors. Trends Pharmacol Sci. 1992;13:61–69.

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