Bioactivity-guided mapping and navigation of chemical space-Reference-Cited by-同舟云学术

Bioactivity-guided mapping and navigation of chemical space

Published:2009-06-28 Issue:8 Volume:5 Page:585-592
ISSN:1552-4450
Container-title:Nature Chemical Biology
language:en
Short-container-title:Nat Chem Biol

Author:

Renner Steffen,van Otterlo Willem A L,Dominguez Seoane Marta,Möcklinghoff Sabine,Hofmann Bettina,Wetzel Stefan,Schuffenhauer Ansgar,Ertl Peter,Oprea Tudor I,Steinhilber Dieter,Brunsveld Luc,Rauh Daniel,Waldmann Herbert

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Molecular Biology

Link

http://www.nature.com/articles/nchembio.188.pdf

Reference30 articles.

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3. Clark, A.M. & Labute, P. Detection and assignment of common scaffolds in project databases of lead molecules. J. Med. Chem. 52, 469–483 (2009).

4. Kaiser, M., Wetzel, S., Kumar, K. & Waldmann, H. Biology-inspired synthesis of compound libraries. Cell. Mol. Life Sci. 65, 1186–1201 (2008).

5. Nören-Müller, A. et al. Discovery of protein phosphatase inhibitor classes by biology-oriented synthesis. Proc. Natl. Acad. Sci. USA 103, 10606–10611 (2006).

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