Enhancing the Small-Scale Screenable Biological Space beyond Known Chemogenomics Libraries with Gray Chemical Matter─Compounds with Novel Mechanisms from High-Throughput Screening Profiles

Author:

Thomas Jason R.1,Shelton Claude1,Murphy Jason1,Brittain Scott1,Bray Mark-Anthony1,Aspesi Peter1,Concannon John1,King Frederick J.2,Ihry Robert J.2ORCID,Ho Daniel J.2,Henault Martin1,Hadjikyriacou Andrea1,Neri Marilisa3,Sigoillot Frederic D.1,Pham Helen T.1,Shum Matthew1,Barys Louise3,Jones Michael D.1,Martin Eric J.4ORCID,Blechschmidt Anke3,Rieffel Sébastien3,Troxler Thomas J.3,Mapa Felipa A.1,Jenkins Jeremy L.1,Jain Rishi K.1,Kutchukian Peter S.1,Schirle Markus1ORCID,Renner Steffen3ORCID

Affiliation:

1. Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States

2. Novartis Biomedical Research, San Diego, California 92121, United States

3. Novartis Biomedical Research, Basel 4056, Switzerland

4. Novartis Biomedical Research, Emeryville, California 94608, United States

Publisher

American Chemical Society (ACS)

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