Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65-Reference-Cited by-同舟云学术

Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65

Published:2015-11 Issue:7579 Volume:527 Page:477-483
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Huang Xi-Ping,Karpiak Joel,Kroeze Wesley K.,Zhu Hu,Chen Xin,Moy Sheryl S.,Saddoris Kara A.,Nikolova Viktoriya D.,Farrell Martilias S.,Wang Sheng,Mangano Thomas J.,Deshpande Deepak A.,Jiang Alice,Penn Raymond B.,Jin Jian,Koller Beverly H.,Kenakin Terry,Shoichet Brian K.,Roth Bryan L.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/nature15699.pdf

Reference59 articles.

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5. Ferguson, F. M. et al. Targeting low-druggability bromodomains: fragment based screening and inhibitor design against the BAZ2B bromodomain. J. Med. Chem. 56, 10183–10187 (2013)

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