Identification of Small-Molecule Antagonists Targeting the Growth Hormone Releasing Hormone Receptor (GHRHR)

Author:

Matsoukas Minos-Timotheos1ORCID,Radomsky Tarryn23,Panagiotopoulos Vasilis1,Preez Robin du23,Papadourakis Michail4,Tsianakas Konstantinos1,Millar Robert P2567,Anderson Ross C23,Spyroulias Georgios A8,Newton Claire L25

Affiliation:

1. University of West Attica, Department of Biomedical Engineering, Athens 12243, Greece

2. Centre for Neuroendocrinology, Department of Immunology, Faculty of Health Sciences, University of Pretoria, Private Bag X323, Gezina, Pretoria 0031, South Africa

3. Department of Physiology, Faculty of Health Sciences, University of Pretoria, Private Bag X323, Gezina, Pretoria 0031, South Africa

4. Cloudpharm PC, Athens 15125, Greece

5. Deanery of Biomedical Sciences, University of Edinburgh, Edinburgh EH8 9JZ, U.K.

6. Institute of Infectious Diseases and Molecular Medicine, Faculty of Health Sciences, University of Cape Town, Cape Town 7925, South Africa

7. School of Medicine, University of St Andrews, St Andrews KY16 9TF, U.K.

8. University of Patras, School of Health Sciences, Department of Pharmacy, University Campus, Rion, Patras 26500, Greece

Funder

State Scholarships Foundation

European Regional Development Fund

Horizon 2020 Framework Programme

South African Medical Research Council

Greece

Publisher

American Chemical Society (ACS)

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