Stereoselective central nervous system effects of the R- and S-isomers of the GABA uptake blocker N -(4,4-di-(3-methylthien-2-yl)but-3-enyl) nipecotic acid in the rat
Author:
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1038/sj.bjp.0702962/fullpdf
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3. GABA transporter heterogeneity: Pharmacology and cellular localization;BORDEN;Neurochem. Int.,1996
4. Tiagabine, SK&F 89976-A, CI-966 and NNC-771 are selective for the cloned GABA uptake transporter GAT-1;BORDEN;Eur. J. Pharmacol. Mol. Pharm.,1994
5. (R)-N-[4,4-Bis(Methyl-2-Thienyl)but-3-en-1-yl]Nipecotic acid binds with high affinity to the brain γ-aminobutyric acid uptake carrier;BRAESTRUP;J. Neurochem.,1990
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