Rapid Method To Determine Intracellular Drug Concentrations in Cellular Uptake Assays: Application to Metformin in Organic Cation Transporter 1-Transfected Human Embryonic Kidney 293 Cells-Reference-Cited by-同舟云学术

Rapid Method To Determine Intracellular Drug Concentrations in Cellular Uptake Assays: Application to Metformin in Organic Cation Transporter 1-Transfected Human Embryonic Kidney 293 Cells

Published:2015-12-23 Issue:3 Volume:44 Page:356-364
ISSN:1521-009X
Container-title:Drug Metabolism and Disposition
language:en
Short-container-title:Drug Metabolism and Disposition

Author:

Chien H.-C.,Zur A. A.,Maurer T. S.,Yee S. W.,Tolsma J.,Jasper P.,Scott D. O.,Giacomini K. M.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmaceutical Science,Pharmacology

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1. Intraluminal calcium as a primary regulator of endoplasmic reticulum function

2. OCT1 is a high-capacity thiamine transporter that regulates hepatic steatosis and is a target of metformin

3. Intracellular Drug Concentrations and Transporters: Measurement, Modeling, and Implications for the Liver

4. Intracellular Drug Concentrations

5. Brain Mitochondrial Drug Delivery: Influence of Drug Physicochemical Properties

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