Design, Synthesis, and Analysis of a Polyethelene Glycol-Modified (PEGylated) Small Molecule Inhibitor of Integrin α4β1 with Improved Pharmaceutical Properties-Reference-Cited by-同舟云学术

Design, Synthesis, and Analysis of a Polyethelene Glycol-Modified (PEGylated) Small Molecule Inhibitor of Integrin α4β1 with Improved Pharmaceutical Properties

Published:2004-10-14 Issue:2 Volume:312 Page:742-750
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Pepinsky R. B.,Lee W.-C.,Cornebise M.,Gill A.,Wortham K.,Chen L. L.,Leone D. R.,Giza K.,Dolinski B. M.,Perper S.,Nickerson-Nutter C.,Lepage D.,Chakraborty A.,Whalley E. T.,Petter R. C.,Adams S. P.,Lobb R. R.,Scott D. M.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference37 articles.

1. Blockade of Late-phase Airway Responses and Airway Hyperresponsiveness in Allergic Sheep with a Small-molecule Peptide Inhibitor of VLA-4

2. Osteopontin is a ligand for the alpha4beta1 integrin

3. Evidence That Ligand and Metal Ion Binding to Integrin α4β1 Are Regulated through a Coupled Equilibrium

4. Integrins and Signal Transduction Pathways: the Road Taken

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