Reversible Inhibitors of Fatty Acid Amide Hydrolase That Promote Analgesia: Evidence for an Unprecedented Combination of Potency and Selectivity-Reference-Cited by-同舟云学术

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Reversible Inhibitors of Fatty Acid Amide Hydrolase That Promote Analgesia: Evidence for an Unprecedented Combination of Potency and Selectivity

Published:2004-06-30 Issue:2 Volume:311 Page:441-448
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Lichtman Aron H.,Leung Donmienne,Shelton Christopher C.,Saghatelian Alan,Hardouin Christophe,Boger Dale L.,Cravatt Benjamin F.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference47 articles.

1. Proteomic profiling of mechanistically distinct enzyme classes using a common chemotype

2. Structure−Function Analysis of Human Triacylglycerol Hydrolase by Site-Directed Mutagenesis: Identification of the Catalytic Triad and a Glycosylation Site

3. Influence of the N-1 alkyl chain length of cannabimimetic indoles upon CB1 and CB2 receptor binding

4. Boger DL, Miyauchi H, Du W, Hardouin C, Fecik RA, Cheng H, Hwang I, Hedrick MP, Leung D, Acevedo O, et al. (2004) Discovery of a potent, selective, and efficacious class of reversible α-ketoheterocycle inhibitors of fatty acid amide hydrolase. J Med Chem, in press.

5. Trifluoromethyl ketone inhibitors of fatty acid amide hydrolase: A probe of structural and conformational features contributing to inhibition

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