Discovery of a Potent, Selective, and Efficacious Class of Reversible α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Effective as Analgesics-Reference-Cited by-同舟云学术

Discovery of a Potent, Selective, and Efficacious Class of Reversible α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Effective as Analgesics

Published:2004-10-23 Issue:6 Volume:48 Page:1849-1856
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Boger Dale L.¹,Miyauchi Hiroshi¹,Du Wu¹,Hardouin Christophe¹,Fecik Robert A.¹,Cheng Heng¹,Hwang Inkyu¹,Hedrick Michael P.¹,Leung Donmienne¹,Acevedo Orlando¹,Guimarães Cristiano R. W.¹,Jorgensen William L.¹,Cravatt Benjamin F.¹

Affiliation:

1. Departments of Chemistry, Cell Biology, and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, and Department of Chemistry, Yale University, 225 Prospect Street, New Haven, Connecticut 06520-8107

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049614v

Reference56 articles.

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