Evaluation of Histamine H1-, H2-, and H3-Receptor Ligands at the Human Histamine H4 Receptor: Identification of 4-Methylhistamine as the First Potent and Selective H4 Receptor Agonist-Reference-Cited by-同舟云学术

Evaluation of Histamine H1-, H2-, and H3-Receptor Ligands at the Human Histamine H4 Receptor: Identification of 4-Methylhistamine as the First Potent and Selective H4 Receptor Agonist

Published:2005-06-09 Issue:3 Volume:314 Page:1310-1321
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Lim Herman D.,van Rijn Richard M.,Ling Ping,Bakker Remko A.,Thurmond Robin L.,Leurs Rob

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference42 articles.

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2. Regulation of human β1-adrenergic receptors and their mRNA in neuroepithelioma SK-N-MC cells: effects of agonist, forskolin, and protein kinase A11Abbreviations: β-AR, β-adrenergic receptor(s); PKA, cyclic AMP-dependent protein kinase A; DMEM, Dulbecco’s modified Eagle’s medium; ICYP, 125I-iodocyanopindolol; PCR, polymerase chain reaction; and GPCR, G protein-coupled receptor

3. Bakker RA (2003) Modulation of Histamine H1-Receptor Activity. Ph.D. Thesis, Vrije Universiteit Amsterdam, The Netherlands.

4. Histamine H1-Receptor Activation of Nuclear Factor-κB: Roles for Gβγ- and Gαq/11-Subunits in Constitutive and Agonist-Mediated Signaling

5. 8R-Lisuride Is a Potent Stereospecific Histamine H1-Receptor Partial Agonist

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