Mutagenesis of Nucleophilic Residues near the Orthosteric Binding Pocket of M1and M2Muscarinic receptors: Effect on the Binding of Nitrogen Mustard Analogs of Acetylcholine and McN-A-343-Reference-Cited by-同舟云学术

Mutagenesis of Nucleophilic Residues near the Orthosteric Binding Pocket of M1and M2Muscarinic receptors: Effect on the Binding of Nitrogen Mustard Analogs of Acetylcholine and McN-A-343

Published:2010-07-19 Issue:4 Volume:78 Page:745-755
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Suga Hinako,Sawyer Gregory W.,Ehlert Frederick J.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference25 articles.

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4. Christopoulos A (2000) Quantification of allosteric interactions at G protein-coupled receptors using radioligand binding assays, in Current Protocols in Pharmacology ( Enna SJ ed) pp 1.22.1–1.22.40, Wiley & Sons, New York.

5. Propylbenzilylcholine mustard labels an acidic residue in transmembrane helix 3 of the muscarinic receptor;Curtis;J Biol Chem,1989

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