Aminergic GPCR–Ligand Interactions: A Chemical and Structural Map of Receptor Mutation Data

Author:

Vass Márton1ORCID,Podlewska Sabina2,de Esch Iwan J. P.1,Bojarski Andrzej J.2ORCID,Leurs Rob1ORCID,Kooistra Albert J.13ORCID,de Graaf Chris14ORCID

Affiliation:

1. Division of Medicinal Chemistry, Faculty of Sciences, Amsterdam Institute for Molecules, Medicines and Systems (AIMMS), VU University Amsterdam, 1081HZ Amsterdam, The Netherlands

2. Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, Smętna 12, PL31-343 Kraków, Poland

3. Department of Drug Design and Pharmacology, University of Copenhagen, Universitetsparken 2, 2100 Copenhagen, Denmark

4. Sosei Heptares, Steinmetz Building, Granta Park, Great Abington, Cambridge CB21 6DG, U.K.

Funder

Narodowe Centrum Nauki

European Cooperation in Science and Technology

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Netherlands eScience Center

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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