RVX-297, a BET Bromodomain Inhibitor, Has Therapeutic Effects in Preclinical Models of Acute Inflammation and Autoimmune Disease-Reference-Cited by-同舟云学术

RVX-297, a BET Bromodomain Inhibitor, Has Therapeutic Effects in Preclinical Models of Acute Inflammation and Autoimmune Disease

Published:2017-09-29 Issue:6 Volume:92 Page:694-706
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Jahagirdar Ravi,Attwell Sarah,Marusic Suzana,Bendele Alison,Shenoy Narmada,McLure Kevin G.,Gilham Dean,Norek Karen,Hansen Henrik C.,Yu Raymond,Tobin Jennifer,Wagner Gregory S.,Young Peter R.,Wong Norman C. W.,Kulikowski Ewelina

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference60 articles.

1. NF-κB is 25

2. Selective inhibition of CD4+ T-cell cytokine production and autoimmunity by BET protein and c-Myc inhibitors

3. Structure of a Domain-Swapped FOXP3 Dimer on DNA and Its Function in Regulatory T Cells

4. I-BET151 selectively regulates IL-6 production

5. Inflammatory bowel disease: cause and immunobiology

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