S1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In Vivo-Reference-Cited by-同舟云学术

S1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In Vivo

Published:2017-12-04 Issue:2 Volume:93 Page:109-118
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Birker-Robaczewska Magdalena,Bolli Martin,Rey Markus,de Kanter Ruben,Kohl Christopher,Lescop Cyrille,Boucher Maxime,Poirey Sylvie,Steiner Beat,Nayler Oliver

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

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4. Amelioration of Collagen-Induced Arthritis by a Novel S1P1Antagonist with Immunomodulatory Activities

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1. Sphingosine 1-phosphate receptor-targeted therapeutics in rheumatic diseases;Nature Reviews Rheumatology;2022-05-04

2. Morpholino Analogues of Fingolimod as Novel and Selective S1P1 Ligands with In Vivo Efficacy in a Mouse Model of Experimental Antigen-Induced Encephalomyelitis;International Journal of Molecular Sciences;2020-09-04

3. Post-translational modifications of S1PR1 and endothelial barrier regulation;Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids;2020-09