Multiple Binding Sites for Small-Molecule Antagonists at the CC Chemokine Receptor 2-Reference-Cited by-同舟云学术

Multiple Binding Sites for Small-Molecule Antagonists at the CC Chemokine Receptor 2

Published:2013-07-22 Issue:4 Volume:84 Page:551-561
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Zweemer Annelien J. M.,Nederpelt Indira,Vrieling Hilde,Hafith Sarah,Doornbos Maarten L. J.,de Vries Henk,Abt Jeffrey,Gross Raymond,Stamos Dean,Saunders John,Smit Martine J.,IJzerman Adriaan P.,Heitman Laura H.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference42 articles.

1. An Intracellular Allosteric Site for a Specific Class of Antagonists of the CC Chemokine G Protein-Coupled Receptors CCR4 and CCR5

2. CCR2: Characterization of the Antagonist Binding Site from a Combined Receptor Modeling/Mutagenesis Approach

3. Delayed Functional Expression of Neuronal Chemokine Receptors Following Focal Nerve Demyelination in the Rat: A Mechanism for the Development of Chronic Sensitization of Peripheral Nociceptors

4. Decreased lesion formation in CCR2−/− mice reveals a role for chemokines in the initiation of atherosclerosis

5. Discovery and Pharmacological Characterization of a Novel Rodent-Active CCR2 Antagonist, INCB3344

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