SSR126768A (4-Chloro-3-[(3R)-(+)-5-chloro-1-(2,4-dimethoxybenzyl)-3-methyl-2- oxo-2,3-dihydro-1H-indol-3-yl]-N-ethyl-N-(3-pyridylmethyl)-benzamide, Hydrochloride): A New Selective and Orally Active Oxytocin Receptor Antagonist for the Prevention of Preterm Labor-Reference-Cited by-同舟云学术

SSR126768A (4-Chloro-3-[(3R)-(+)-5-chloro-1-(2,4-dimethoxybenzyl)-3-methyl-2- oxo-2,3-dihydro-1H-indol-3-yl]-N-ethyl-N-(3-pyridylmethyl)-benzamide, Hydrochloride): A New Selective and Orally Active Oxytocin Receptor Antagonist for the Prevention of Preterm Labor

Published:2004-01-13 Issue:1 Volume:309 Page:414-424
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Serradeil-Le Gal Claudine,Valette Gérard,Foulon Loïc,Germain Guy,Advenier Charles,Naline Emmanuel,Bardou Marc,Martinolle Jean-Pierre,Pouzet Brigitte,Raufaste Danielle,Garcia Corinne,Double-Cazanave Eléonore,Pauly Maxime,Pascal Marc,Barbier Alain,Scatton Bernard,Maffrand Jean-Pierre,Le Fur Gérard

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference40 articles.

1. Chapter 28 Involvement of oxytocin and vasopressin in the pathophysiology of preterm labor and primary dysmenorrhea

2. Receptor binding of oxytocin and vasopressin antagonists and inhibitory effects on isolated myometrium from preterm and term pregnant women

3. Inhibition of uterine contractions of premature labour with an oxytocin analogue. Results from a pilot study

4. Allen MJ, Smith J, Hampton S, and Giles H (1997) Affinity of antagonists and endogenous peptides at human recombinant oxytocin and vasopressin receptors, in Word Congress of Neurohypophysial Hormones, Montreal, Canada, August 8-12, A176 (Abstr.)

Cited by 53 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Development and validation of CYP26A1 inhibition assay for high‐throughput screening;Biotechnology Journal;2024-06

2. Oxytocin and vasopressin signaling in health and disease;Trends in Biochemical Sciences;2024-04

3. Enantioselective Nucleophilic Vinylic Substitution (S_NV) toward 3-Alkenyl-bisoxindoles Facilitated by C6′ Steric Bulk of Cinchona Alkaloid;Organic Letters;2023-08-03

4. THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors;British Journal of Pharmacology;2021-09-16

5. Oxytocin in the Male Reproductive Tract; The Therapeutic Potential of Oxytocin-Agonists and-Antagonists;Frontiers in Endocrinology;2020-10-22