Discovery and Mapping of an Intracellular Antagonist Binding Site at the Chemokine Receptor CCR2-Reference-Cited by-同舟云学术

Discovery and Mapping of an Intracellular Antagonist Binding Site at the Chemokine Receptor CCR2

Published:2014-07-14 Issue:4 Volume:86 Page:358-368
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Zweemer Annelien J.M.,Bunnik Julia,Veenhuizen Margo,Miraglia Fabiana,Lenselink Eelke B.,Vilums Maris,de Vries Henk,Gibert Arthur,Thiele Stefanie,Rosenkilde Mette M.,IJzerman Adriaan P.,Heitman Laura H.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference49 articles.

1. An Intracellular Allosteric Site for a Specific Class of Antagonists of the CC Chemokine G Protein-Coupled Receptors CCR4 and CCR5

2. [19] Integrated methods for the construction of three-dimensional models and computational probing of structure-function relations in G protein-coupled receptors

3. Decreased lesion formation in CCR2−/− mice reveals a role for chemokines in the initiation of atherosclerosis

4. Discovery and Pharmacological Characterization of a Novel Rodent-Active CCR2 Antagonist, INCB3344

5. Nonpeptidergic Allosteric Antagonists Differentially Bind to the CXCR2 Chemokine Receptor

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