Development of a Fluorescent Ligand for the Intracellular Allosteric Binding Site of the Neurotensin Receptor 1-Reference-Cited by-同舟云学术

Development of a Fluorescent Ligand for the Intracellular Allosteric Binding Site of the Neurotensin Receptor 1

Published:2024-04-18 Issue:5 Volume:7 Page:1533-1545
ISSN:2575-9108
Container-title:ACS Pharmacology & Translational Science
language:en
Short-container-title:ACS Pharmacol. Transl. Sci.

Author:

Vogt Hannah¹,Shinkwin Patrick¹,Huber Max E.¹,Staffen Nico¹,Hübner Harald¹,Gmeiner Peter¹²,Schiedel Matthias¹³,Weikert Dorothee¹²

Affiliation:

1. Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander-Universität Erlangen-Nürnberg, Nikolaus-Fiebiger-Straße 10, 91058 Erlangen, Germany

2. FAU NeW − Research Center New Bioactive Compounds, Friedrich-Alexander-Universität Erlangen-Nürnberg, Nikolaus-Fiebiger-Str. 10, 91058 Erlangen, Germany

3. Institute of Medicinal and Pharmaceutical Chemistry, Technische Universität Braunschweig, Beethovenstraße 55, 38106 Braunschweig, Germany

Funder

Deutsche Forschungsgemeinschaft

Verband der Chemischen Industrie

Dr. Hertha und Helmut Schmauser-Stiftung

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acsptsci.4c00086

Reference55 articles.

1. Structural diversity of G protein-coupled receptors and significance for drug discovery

2. G Protein-Coupled Receptors as Targets for Approved Drugs: How Many Targets and How Many Drugs?

3. Delivery of peptide and protein drugs over the blood–brain barrier

4. Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders

5. Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors

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