INFLUX AND EFFLUX TRANSPORT OF H1-ANTAGONIST EPINASTINE ACROSS THE BLOOD-BRAIN BARRIER-Reference-Cited by-同舟云学术

INFLUX AND EFFLUX TRANSPORT OF H1-ANTAGONIST EPINASTINE ACROSS THE BLOOD-BRAIN BARRIER

Published:2004-04-20 Issue:5 Volume:32 Page:519-524
ISSN:0090-9556
Container-title:Drug Metabolism and Disposition
language:en
Short-container-title:Drug Metab Dispos

Author:

Ishiguro Naoki,Nozawa Takashi,Tsujihata Akiko,Saito Asami,Kishimoto Wataru,Yokoyama Kazutoshi,Yotsumoto Takafumi,Sakai Kenji,Igarashi Takashi,Tamai Ikumi

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmaceutical Science,Pharmacology

Reference29 articles.

1. Antihistamine activity and central effects of WAL 801 CL in man

2. Blood-Brain Barrier Is Involved in the Efflux Transport of a Neuroactive Steroid, Dehydroepiandrosterone Sulfate, via Organic Anion Transporting Polypeptide 2

3. P-Glycoprotein Limits the Brain Penetration of Nonsedating but not Sedating H1-Antagonists

4. Affinity for the P-Glycoprotein Efflux Pump at the Blood-Brain Barrier May Explain the Lack of CNS Side-Effects of Modern Antihistamines

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Characterization of Aripiprazole Uptake Transporter in the Blood-Brain Barrier Model hCMEC/D3 Cells by Targeted siRNA Screening;Pharmaceutical Research;2022-03-21

2. Prediction of negative food effect induced by bile micelle binding on oral absorption of hydrophilic cationic drugs;European Journal of Pharmaceutical Sciences;2020-12

3. Simultaneous measurement of epinastine and its metabolite, 9,13b‐dehydroepinastine, in human plasma by a newly developed ultra‐performance liquid chromatography–tandem mass spectrometry and its application to pharmacokinetic studies;Biomedical Chromatography;2020-06-25

4. Cell-based, animal and H1 receptor binding studies relative to the sedative effects of ketotifen and norketotifen atropisomers;Journal of Pharmacy and Pharmacology;2020-02-06

5. Using miniature brain implants in rodents for novel drug discovery;Expert Opinion on Drug Discovery;2019-03-04