Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit β-Arrestin-2

Author:

Váradi András1,Marrone Gina F.1,Palmer Travis C.1,Narayan Ankita1,Szabó Márton R.2,Le Rouzic Valerie1,Grinnell Steven G.1,Subrath Joan J.1,Warner Evelyn1,Kalra Sanjay1,Hunkele Amanda1,Pagirsky Jeremy1,Eans Shainnel O.3,Medina Jessica M.3,Xu Jin1,Pan Ying-Xian1,Borics Attila2,Pasternak Gavril W.1,McLaughlin Jay P.3,Majumdar Susruta1

Affiliation:

1. Molecular Pharmacology and Chemistry Program and Department of Neurology, Memorial Sloan Kettering Cancer Center, New York, New York 10065, United States

2. Institute of Biochemistry, Biological Research Centre, Hungarian Academy of Sciences, Szeged, H-6726 Hungary

3. Department of Pharmacodyanamics, University of Florida, Gainesville, Florida 032610, United States

Funder

National Cancer Institute

Magyar Tudományos Akadémia

Division of Graduate Education

National Institute on Drug Abuse

Office of Tourism, Trade, and Economic Development, State of Florida

Peter F. McManus Charitable Trust

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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