Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists-Reference-Cited by-同舟云学术

Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists

Published:2016-04-05 Issue:7 Volume:59 Page:3452-3470
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Geyer Roland¹,Nordemann Uwe¹,Strasser Andrea¹,Wittmann Hans-Joachim¹,Buschauer Armin¹

Affiliation:

1. Institute of Pharmacy, Pharmaceutical/Medicinal Chemistry, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b00120

Reference89 articles.

1. Discovery of a Novel Member of the Histamine Receptor Family

2. Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in Leukocytes

3. Molecular Cloning and Characterization of a New Human Histamine Receptor, HH4R

4. Cloning, Expression, and Pharmacological Characterization of a Novel Human Histamine Receptor

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