Biological Characterization and in Vivo Assessment of the Activity of a New Synthetic Macrocyclic Antifungal Compound

Author:

Deodato Davide12,Maccari Giorgio12,De Luca Filomena3,Sanfilippo Stefania1,Casian Alexandru1,Martini Riccardo1,D’Arezzo Silvia4,Bonchi Carlo5,Bugli Francesca6,Posteraro Brunella7,Vandeputte Patrick8,Sanglard Dominique8,Docquier Jean-Denis32,Sanguinetti Maurizio67,Visca Paolo5,Botta Maurizio192

Affiliation:

1. Department of Biotechnology Chemistry and Pharmacy, University of Siena, I-53100 Siena, Italy

2. Lead Discovery Siena s.r.l., Via Vittorio Alfieri 31, I-53019 Castelnuovo Berardenga, Italy

3. Department of Medical Biotechnology, University of Siena, I-53100 Siena, Italy

4. Istituto Nazionale per le Malattie Infettive “Lazzaro Spallanzani”, I-00149 Roma, Italy

5. Dipartimento di Scienze, Università Roma Tre, I-00154 Roma, Italy

6. Institute of Microbiology, Università Cattolica del Sacro Cuore, I-00168 Roma, Italy

7. Institute of Public Health, Università Cattolica del Sacro Cuore, I-00168 Roma, Italy

8. Institute of Microbiology, University of Lausanne and University Hospital Center, CH-1011 Lausanne, Switzerland

9. Sbarro Institute for Cancer Research and Molecular Medicine, Temple University, BioLife Science Building, Suite 333, 1900 North 12th Street, Philadelphia, Pennsylvania 19122, United States,

Funder

Swiss National Science Foundation

Bakker Medical Srl

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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