Targeting the Non-Catalytic Functions: a New Paradigm for Kinase Drug Discovery?

Author:

Wang Zhen1ORCID,Huang Weixue1,Zhou Kaijie1,Ren Xiaomei2,Ding Ke1234ORCID

Affiliation:

1. State Key Laboratory of Bioorganic and Natural Products Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, #345 Ling Ling Road, Shanghai 200032, People’s Republic of China

2. International Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Development, Ministry of Education (MoE) of People’s Republic of China, College of Pharmacy, Jinan University, 601 Huangpu Avenue West, Guangzhou 510632, People’s Republic of China

3. The First Affiliated Hospital (Huaqiao Hospital), Jinan University, 601 Huangpu Avenue West, Guangzhou 510632, People’s Republic of China

4. Institute of Basic Medicine and Cancer (IBMC), Chinese Academy of Sciences, Hangzhou, Zhejiang 310022, People’s Republic of China

Funder

State Key Laboratory of Bio-organic and Natural Products Chemistry

National Natural Science Foundation of China

Open Project of Shenzhen Bay Laboratory

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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