Melanocortin 1 Receptor Agonists Based on a Bivalent, Bicyclic Peptide Framework-Reference-Cited by-同舟云学术

Melanocortin 1 Receptor Agonists Based on a Bivalent, Bicyclic Peptide Framework

Published:2021-07-01 Issue:14 Volume:64 Page:9906-9915
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Durek Thomas¹^ORCID,Kaas Quentin¹^ORCID,White Andrew M.¹^ORCID,Weidmann Joachim¹,Fuaad Abdullah Ahmad¹,Cheneval Olivier¹^ORCID,Schroeder Christina I.¹^ORCID,de Veer Simon J.¹^ORCID,Dellsén Anita²,Österlund Torben³⁴,Larsson Niklas³,Knerr Laurent⁵^ORCID,Bauer Udo⁵,Plowright Alleyn T.⁵,Craik David J.¹^ORCID

Affiliation:

1. Institute for Molecular Bioscience, Australian Research Council Centre of Excellence for Innovations in Peptide and Protein Science, The University of Queensland, Brisbane, QLD 4072, Australia

2. Mechanistic Biology & Profiling, Discovery Sciences, IMED Biotech Unit, AstraZeneca, Gothenburg 43183, Mölndal, Sweden

3. Discovery Biology, Discovery Sciences, IMED Biotech Unit, AstraZeneca, Gothenburg 43183, Mölndal, Sweden

4. Drug Safety and Metabolism, IMED Biotech Unit, AstraZeneca, Gothenburg 43183, Mölndal, Sweden

5. Medicinal Chemistry, Cardiovascular and Metabolic Diseases, IMED Biotech Unit, AstraZeneca, Gothenburg 43183, Mölndal, Sweden

Funder

National Health and Medical Research Council

Australian Research Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00095

Reference40 articles.

1. The Melanocortin Receptor System: A Target for Multiple Degenerative Diseases

2. MOLECULAR EVOLUTION OF GPCRS: Melanocortin/melanocortin receptors

3. Intracellular signaling mechanisms of the melanocortin receptors: current state of the art

4. .alpha.-Melanotropin: the minimal active sequence in the frog skin bioassay

5. Determination of the melanocortin-4 receptor structure identifies Ca 2+ as a cofactor for ligand binding

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