Discovery of Potent and Fast-Acting Antimalarial Bis-1,2,4-triazines-Reference-Cited by-同舟云学术

Discovery of Potent and Fast-Acting Antimalarial Bis-1,2,4-triazines

Published:2021-03-24 Issue:7 Volume:64 Page:4150-4162
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Priebbenow Daniel L.¹^ORCID,Mathiew Mitch²,Shi Da-Hua²,Harjani Jitendra R.²,Beveridge Julia G.²,Chavchich Marina³,Edstein Michael D.³,Duffy Sandra,Avery Vicky M.,Jacobs Robert T.⁴,Brand Stephen⁴,Shackleford David M.⁵,Wang Wen⁵,Zhong Longjin⁵,Lee Given⁵,Tay Erin⁵,Barker Helena⁵,Crighton Elly⁵,White Karen L.⁵,Charman Susan A.⁵,De Paoli Amanda⁶,Creek Darren J.⁶^ORCID,Baell Jonathan B.²⁷^ORCID

Affiliation:

1. School of Chemistry, The University of Melbourne, Parkville, VIC 3010, Australia

2. Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), 381 Royal Parade, Parkville, VIC 3052, Australia

3. The Department of Drug Evaluation, Australian Defence Force Malaria and Infectious Disease Institute, Brisbane, QLD 4051, Australia

4. Medicines for Malaria Venture (MMV), P.O. Box 1826, Route de Pré-Bois 20, CH-1215 Geneva, Switzerland

5. Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), 381 Royal Parade, Parkville, VIC 3052, Australia

6. Drug Delivery Disposition and Dynamics, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), 381 Royal Parade, Parkville, VIC 3052, Australia

7. ARC Centre for Fragment-Based Design, Monash University (Parkville Campus), 381 Royal Parade, Parkville, VIC 3052, Australia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00044

Reference35 articles.

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2. Malaria

3. Recent updates in the discovery and development of novel antimalarial drug candidates

4. Triazolopyrimidine-Based Dihydroorotate Dehydrogenase Inhibitors with Potent and Selective Activity against the Malaria Parasite Plasmodium falciparum

5. Lead Optimization of Aryl and Aralkyl Amine-Based Triazolopyrimidine Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase with Antimalarial Activity in Mice

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