Targeting a Novel KRAS Binding Site: Application of One-Component Stapling of Small (5–6-mer) Peptides
Author:
Affiliation:
1. Department of Chemistry, Cambridge University, Lensfield Road, Cambridge CB2 1EW, U.K.
2. Chemistry, Oncology R&D, AstraZeneca, Cambridge CB4 0WG, U.K.
3. Discovery Sciences, BioPharmaceuticals R&D, AstraZeneca, Cambridge CB4 0WG, U.K.
Funder
AstraZeneca
Engineering and Physical Sciences Research Council
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01334
Reference45 articles.
1. PKC Regulates a Farnesyl-Electrostatic Switch on K-Ras that Promotes its Association with Bcl-Xl on Mitochondria and Induces Apoptosis
2. Roles of the Ras/Raf/MEK/ERK pathway in leukemia therapy
3. Dragging Ras Back in the Ring
4. A Comprehensive Survey of Ras Mutations in Cancer
5. Targeting RAS signalling pathways in cancer therapy
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