Accelerated Identification of Cell Active KRAS Inhibitory Macrocyclic Peptides using Mixture Libraries and Automated Ligand Identification System (ALIS) Technology
Author:
Affiliation:
1. Merck & Co., Inc., Boston, Massachusetts 02115, United States
2. MSD International, Singapore 138665, Singapore
3. Merck & Co., Inc., Kenilworth, New Jersey 07033, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00154
Reference42 articles.
1. Drugging the undruggable RAS: Mission Possible?
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5. Cracking KRAS
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